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Novel isoxazole thiophene-containing compounds active against Mycobacterium tuberculosis

Gabrielle Martinez1, Kirsten Tolentino1, Paridhi Sukheja1

  • 1Calibr-Skaggs Institute for Innovative Medicines, a division of Scripps Research, La Jolla, CA 92037, United States.

Bioorganic & Medicinal Chemistry Letters
|January 25, 2025
PubMed

Keywords:
CholesterolCytotoxicityFormal hit profilingHit to leadMycobacterium tuberculosisPharmacokineticRv1625c/CyaStructure–activity relationship

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