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Updated: May 28, 2025

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
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A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators

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Covalent-Allosteric Inhibitors: Do We Get the Best of Both Worlds?

Hui Tao1, Bo Yang1, Atena Farhangian1

  • 1Borch Department of Medicinal Chemistry and Molecular Pharmacology, Purdue Institute for Drug Discovery, Purdue University, West Lafayette, Indiana 47907, United States.

Journal of Medicinal Chemistry
|February 12, 2025
PubMed

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