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Updated: May 27, 2025

Facile Preparation of 2Z,4E-Dienamides by the Olefination of Electron-deficient Alkenes with Allyl Acetate
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Use of Aldehyde-Alkyne-Amine Couplings to Generate Medicinal Chemistry-Relevant Linkers

Andrew McGown1, Vesna Vetma2, Damien Crepin1

  • 1Sussex Drug Discovery Centre, School of Life Sciences, University of Sussex, Falmer BN1 9QJ, U.K.

ACS Medicinal Chemistry Letters
|February 19, 2025
PubMed

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