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Updated: May 23, 2025

A Method for Screening and Validation of Resistant Mutations Against Kinase Inhibitors
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Pyrazolopyrimidines: A Promising Frontier in Cancer Treatment-Reviewing Their Potential as Inhibitors of

Ahmed M Abdelhamed1, Amira A Helwa1, Hanan H Kadry2

  • 1Pharmaceutical Organic Chemistry Department, College of Pharmaceutical Sciences and Drug Manufacturing, Misr University for Science and Technology (MUST), 6th of October City, Egypt.

Chemistry & Biodiversity
|March 10, 2025
PubMed

Keywords:
ATP‐binding sitekinase inhibitionpyrazolopyrimidine derivativesserine/threonine kinasestructure–activity relationship

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