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Updated: May 22, 2025

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A Direct, Regioselective and Atom-Economical Synthesis of 3-Aroyl-N-hydroxy-5-nitroindoles by Cycloaddition of 4-Nitronitrosobenzene with Alkynones

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Silver-Catalyzed and Base-Mediated Double Cyclization for the Streamlined Synthesis of

Kanokwan Jaithum1, Jumreang Tummatorn1,2, Chatphorn Theppitak2

  • 1Program on Chemical Sciences, Center of Excellence on Environmental Health and Toxicology (EHT), OPS, MHESI, Chulabhorn Graduate Institute, 54 Kamphaeng Phet 6, Laksi, Bangkok, 10210, Thailand.

Chemistry, an Asian Journal
|March 13, 2025
PubMed

Keywords:
BenzoimidazoleDouble cyclizationNaphthooxazoleOrtho‐‐AlkynylarylketonesSilver catalyst

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