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Novel Pyrimidinyl Sulfonamide Derivatives as GPR17 Modulators

Taoqian Zhao1, Steven H Liang1

  • 1Department of Radiology and Imaging Sciences, Emory University, Atlanta, Georgia 30322, United States.

ACS Medicinal Chemistry Letters
|March 19, 2025
PubMed
Summary

Novel pyrimidinyl sulfonamide derivatives were developed to modulate GPR17 activities. These compounds show promise for treating diseases linked to GPR17 antagonism.

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