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Design, synthesis, and biological evaluation of hypoxic-activation prodrug TH-302 derivatives

Zhengyi Li1, Xingchen Yang1, Shun Wang1

  • 1Jiangsu Key Laboratory of Advanced Catalytic Materials & Technology, School of Petrochemical Engineering, Changzhou University, Changzhou, Jiangsu 213164, China.

Bioorganic & Medicinal Chemistry Letters
|March 19, 2025
PubMed

Keywords:
Anticancer activityGlioblastomaHypoxia-activated prodrugOvarian cancerTH-302 derivatives

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