Exploiting structural variability in the kinase back-pocket to modulate polypharmacology of TAM inhibitors

Megan D Hopkins1, Dehui Zhang1, Zhilong Chen1

  • 1Center for Integrative Chemical Biology and Drug Discovery, Division of Chemical Biology and Medicinal Chemistry, Eshelman School of Pharmacy, University of North Carolina at Chapel Hill, Chapel Hill, NC 27599, USA.

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