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Updated: May 13, 2025

Protein WISDOM: A Workbench for In silico De novo Design of BioMolecules
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Design, Synthesis, and Biological Implications of Autotaxin inhibitors with a Three-Point lock binding mode

Nicolas Desroy1, Razvan Borza2, Jörg Heiermann3

  • 1Galapagos SASU, 102 Avenue Gaston Roussel, 93230 Romainville, France.

Bioorganic & Medicinal Chemistry
|April 15, 2025
PubMed

Keywords:
AutotaxinAutotaxin inhibitorCrystal structureImidazo[12–b]pyridazineLysophosphatidic acidZinc binder

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