PDZK1 inhibits MRP2-mediated oxaliplatin chemosensitivity in hepatocellular carcinoma

Zeqi Duan1, Jinyu Li2,3, Chao Ren4

  • 1First Clinical Medical College, Shanxi Medical University, Taiyuan, 030001, Shanxi Province, People's Republic of China.

Scientific Reports
|April 18, 2025
PubMed

Insights

High PDZK1 expression predicts poor prognosis and oxaliplatin resistance in hepatocellular carcinoma (HCC). PDZK1 enhances HCC cell growth by activating the MRP2-mediated pathway, suggesting it as a biomarker for oxaliplatin chemotherapy sensitivity.

Area of Science:

  • Oncology
  • Molecular Biology
  • Biochemistry

Background:

  • Recurrence following oxaliplatin (OXA) chemotherapy presents a significant challenge for advanced hepatocellular carcinoma (HCC) patients.
  • Identifying biomarkers for OXA-treated recurrence is crucial for improving patient outcomes.

Purpose of the Study:

  • To investigate the role of PDZK1 in oxaliplatin resistance and prognosis in hepatocellular carcinoma.
  • To elucidate the underlying molecular mechanisms involving PDZK1 and MRP2 in HCC chemosensitivity.

Main Methods:

  • Differential gene expression analysis and Kaplan-Meier survival analysis using public databases (GSE51951, TCGA-LIHC, Chinese Liver Cancer Atlas).
  • Retrospective analysis of 39 HCC cases treated with platinum-based drugs.
  • Immunohistochemistry, cell culture models, subcutaneous tumor models, Gene Set Enrichment Analysis (GSEA), Co-Immunoprecipitation (Co-IP), and immunofluorescence assays.

Main Results:

  • High PDZK1 expression correlated with OXA resistance and poor prognosis in HCC.
  • PDZK1 overexpression promoted HCC cell viability, migration, and invasion in vitro and in vivo following OXA treatment.
  • PDZK1 interacted with and co-localized with MRP2, activating MRP2-mediated ABC transporter and bile acid metabolism pathways.
  • Clinical specimens showed a positive correlation between PDZK1 and MRP2 protein levels.

Conclusions:

  • PDZK1 is a novel biomarker associated with oxaliplatin chemosensitivity in HCC.
  • PDZK1 enhances OXA sensitivity in HCC by activating the MRP2-mediated signaling pathway, offering a potential therapeutic target.

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