Enhancing Transthyretin Binding Affinity Prediction with a Consensus Model: Insights from the Tox24 Challenge

Xiaolin Pan1, Yaowen Gu1, Weijun Zhou1

  • 1Department of Chemistry, New York University, New York, New York 10003, United States.

PubMed

Insights

This study developed a deep learning consensus model to predict transthyretin (TTR) binding affinity, integrating multiple molecular data types. The model achieved high accuracy, demonstrating its potential for identifying toxic compounds and assessing endocrine disruption risks.

Area of Science:

  • Computational chemistry
  • Toxicology
  • Molecular modeling

Background:

  • Transthyretin (TTR) is crucial for thyroid hormone transport and homeostasis.
  • Exogenous compounds interacting with TTR can disrupt endocrine function and cause toxicity.

Purpose of the Study:

  • To develop a deep learning-based consensus model for predicting TTR binding affinity.
  • To evaluate the model's performance in the Tox24 challenge and assess its utility for identifying potential TTR binders.

Main Methods:

  • Integrated three deep learning models (sPhysNet, KANO, GGAP-CPI) utilizing 2D, 3D, and protein-ligand interaction data.
  • Developed a consensus model for enhanced predictive accuracy of TTR binding affinity.
  • Utilized the standard deviation of ensemble outputs as an uncertainty estimate for predictions.

Main Results:

  • The consensus model achieved an RMSE of 20.8 on the blind test set, ranking fifth in the Tox24 challenge.
  • Incorporating additional data reduced the RMSE to 20.6 in a retrospective study.
  • Prediction error and RMSE increased with model uncertainty, validating uncertainty as a confidence measure.

Conclusions:

  • Combining regression models across different modalities significantly improves predictive accuracy for TTR binding affinity.
  • The developed consensus model is a valuable tool for in silico prediction of TTR binders and their affinities.
  • Uncertainty estimation provides a reliable measure of prediction confidence, aiding in risk assessment.

Related Concept Videos

Predicting Molecular Geometry02:27

Predicting Molecular Geometry

VSEPR Theory for Determination of Electron Pair Geometries
Relative Strengths of Conjugate Acid-Base Pairs02:29

Relative Strengths of Conjugate Acid-Base Pairs

Brønsted-Lowry acid-base chemistry is the transfer of protons; thus, logic suggests a relation between the relative strengths of conjugate acid-base pairs. The strength of an acid or base is quantified in its ionization constant, Ka or Kb, which represents the extent of the acid or base ionization reaction. For the conjugate acid-base pair HA / A−, the ionization equilibrium equations and ionization constant expressions are
Common Ion Effect03:24

Common Ion Effect

Compared with pure water, the solubility of an ionic compound is less in aqueous solutions containing a common ion (one also produced by dissolution of the ionic compound). This is an example of a phenomenon known as the common ion effect, which is a consequence of the law of mass action that may be explained using Le Châtelier’s principle. Consider the dissolution of silver iodide:
Predicting Reaction Outcomes02:24

Predicting Reaction Outcomes

Kinetics describes the rate and path by which a reaction occurs. In contrast, thermodynamics deals with state functions and describes the properties, behavior, and components of a system. It is not concerned with the path taken by the process and cannot address the rate at which a reaction occurs. Although it does provide information about what can happen during a reaction process, it does not describe the detailed steps of what appears on an atomic or a molecular level. On the other hand,...
Toxic Reactions: Overview01:26

Toxic Reactions: Overview

When toxic substances penetrate the human body, they disseminate to various tissues, undergoing metabolic changes. This process yields reactive metabolites that may covalently bind with specific target molecules, resulting in toxicity.
Toxicity falls into two primary categories: local and systemic.
Local toxicity appears at the exposure site, such as protein denaturation caused by caustic substances.
In contrast, systemic toxicity requires the toxic agent's absorption and distribution,...
Parameters Affecting Nonlinear Elimination: Zero-Order Input, First-Order Absorption and Two-Compartment Model01:13

Parameters Affecting Nonlinear Elimination: Zero-Order Input, First-Order Absorption and Two-Compartment Model

Drugs administered through various routes can lead to nonlinear elimination, resulting in complex pharmacokinetic behaviors crucial to understanding efficacious drug dosing.
When a drug is administered through a constant intravenous infusion and eliminated via nonlinear pharmacokinetics, it follows zero-order input. For example, oral drugs undergo first-order absorption upon administration and are eliminated through nonlinear pharmacokinetics.
In the case of subcutaneously administered drugs,...