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Updated: Jun 13, 2025

A Method for Screening and Validation of Resistant Mutations Against Kinase Inhibitors
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A Method for Screening and Validation of Resistant Mutations Against Kinase Inhibitors

Published on: December 7, 2014

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Discovery of KIN-8741, a Highly Selective Type IIb c-Met Kinase Inhibitor with Broad Mutation Coverage and Quality

Xiaohu S Ouyang1, Kathryn B Grandinetti1, Morgan Boren1

  • 1Kinnate Biopharma Inc., San Diego, California 92130, United States.

Journal of Medicinal Chemistry
|June 3, 2025
PubMed

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