Related Experiment Video

Updated: Jun 15, 2025

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
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A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators

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Multiple intramolecular triggers converge to preferential G protein coupling in the CB2R

Adrian Morales-Pastor1, Tamara Miljuš2,3,4,5,6, Miguel Dieguez-Eceolaza1

  • 1Research Programme on Biomedical Informatics, Hospital del Mar Research Institute and Department of Medicine and Life Science, Universitat Pompeu Fabra, Barcelona, Spain.

Nature Communications
|June 11, 2025
PubMed
Abstract

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