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HTS Identifies NUP98-KDM5A-PHD3 Domain Ligands with Novel Scaffolds

Wenwei Lin1, P Jake Slavish1, Aaron H Phillips1

  • 1†Department of Chemical Biology and Therapeutics, ‡Department of Structural Biology, and §Department of Pathology, St. Jude Children's Research Hospital, Memphis, Tennessee 38105, United States.

ACS Medicinal Chemistry Letters
|June 25, 2025
PubMed

Keywords:
H3K4Me3HTSNUP98-KDM5A PHD3TR-FRET

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