One-pot synthesis of trans-2,3-diaminoindolines through 2,3-diamination of electrophilic indolines

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A Direct, Regioselective and Atom-Economical Synthesis of 3-Aroyl-N-hydroxy-5-nitroindoles by Cycloaddition of 4-Nitronitrosobenzene with Alkynones
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A Direct, Regioselective and Atom-Economical Synthesis of 3-Aroyl-N-hydroxy-5-nitroindoles by Cycloaddition of 4-Nitronitrosobenzene with Alkynones

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Yuito Kobori1, Keisuke Tokushige1, Takumi Abe1

  • 1Graduate School of Medicine, Dentistry and Pharmaceutical Sciences, Okayama University, 1-1-1 Tsushima-naka, Kita-ku, Okayama 7008530, Japan. t-abe@okayama-u.ac.jp.

Organic & Biomolecular Chemistry
|July 2, 2025
PubMed

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