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Small-molecule Cathepsin K inhibitors: a medicinal chemistry perspective

Xuan Guan1,2, Shu Cheng1, Yifei Yin1

  • 1State Key Laboratory of Oral Diseases, West China School of Stomatology, National Clinical Research Center for Oral Diseases, Sichuan University, Chengdu, China.

Future Medicinal Chemistry
|August 5, 2025
PubMed
Abstract

Keywords:
Cathepsin Kdrug designmolecular binding modessmall molecule inhibitorsstructure-activity relationships (SAR)

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