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Updated: Sep 10, 2025

Development of Inhibitors of Protein-protein Interactions through REPLACE: Application to the Design and Development Non-ATP Competitive CDK Inhibitors
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Development of Inhibitors of Protein-protein Interactions through REPLACE: Application to the Design and Development Non-ATP Competitive CDK Inhibitors

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CREB binding protein (CREBBP): Structure-based perspectives for the development of clinical inhibitors

Rongxing Liu1, Jiaxin Li1, Qing Nian2

  • 1Department of Pharmacy, The Second Affiliated Hospital of Army Medical University, 83 Xinqiao Road, Shapingba, Chongqing, China.

Translational Oncology
|August 19, 2025
PubMed

Keywords:
AcetylationCBPInhibitorStructure

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