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Desulfinative Cross-Coupling as a Method to Overcome Problematic Suzuki-Miyaura Reactions of Pharmaceutically

David C Blakemore1, Andre Shavnya1, Michael C Willis2

  • 1Medicine Design, Pfizer Inc., Groton, Connecticut 06340, United States.

ACS Medicinal Chemistry Letters
|August 20, 2025
PubMed

Keywords:
cross-couplingdesulfinativeheterocycleparallel synthesispyridinesulfinatesulfone

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