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Formal synthesis of a selective estrogen receptor modulator with tetrahydrofluorenone structure using [3 + 2 + 1]

Jing Zhang1, Guanyu Zhang2, Hongxi Bai2

  • 1Pingshan Translational Medicine Center, Shenzhen Bay Laboratory, Shenzhen, 518118, China.

Beilstein Journal of Organic Chemistry
|August 21, 2025
PubMed

Keywords:
[3 + 2 + 1] cycloadditionselective estrogen receptor modulatorssynthesistetrahydrofluorenone

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