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Genetically-encoded Molecular Probes to Study G Protein-coupled Receptors
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Structure-Encoded Location Biased Signaling in a Class B GPCR: Focus on the PTH Type 1 Receptor

Karina A Peña1, Jean-Pierre Vilardaga2,3

  • 1Department of Pharmacology and Chemical Biology, University of Pittsburgh School of Medicine, Pittsburgh, PA, USA.

Handbook of Experimental Pharmacology
|September 9, 2025
PubMed

Keywords:
Biased ligandEndosomal signalingG protein-coupled receptorLocation bias signalingParathyroid hormoneStructural dynamics

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