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Updated: Jan 16, 2026

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Structural Perspectives on Biased Allostery of GPCR Signaling

Chang Zhao1,2, Siyuan Shen1, Chao Wu1,2

  • 1Division of Nephrology and Kidney Research Institute, State Key Laboratory of Biotherapy and Cancer Center, West China Hospital, Sichuan University, Chengdu, China.

Handbook of Experimental Pharmacology
|October 1, 2025
PubMed

Keywords:
Allosteric modulatorBiased allosteryBiased signalingMolecular mechanismPharmacology

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