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Characterization of Membrane Transporters by Heterologous Expression in E. coli and Production of Membrane Vesicles
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Cooperativity between endogenous glutamylcysteinylglycine-based oligopeptides and drugs determines the function of

Katja Stefan1, Muhammad Rafehi2, Hauke Busch3

  • 1University of Lübeck and University Medical Center Schleswig-Holstein, Lübeck Institute of Experimental Dermatology, Medicinal Chemistry and Systems Polypharmacology, Ratzeburger Allee 160, 23538 Lübeck, Germany; University of Oslo and Oslo University Hospital, Department of Pathology, Rikshospitalet, Sognsvannsveien 20, 0372 Oslo, Norway.

Biochemical Pharmacology
|October 14, 2025
PubMed

Keywords:
ABC transporterATPaseActivatorMDRMRP1Multidrug resistanceNon-essential activation

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