Histone H3 Lysine 18 Lactylation Promotes Cardiac Hypertrophy Through Activating GATA Binding Protein 4 Signaling

Mingzhu Wang1, Zixian Liu1, Yongbo Ma1

  • 1Yueyang Hospital of Integrated Traditional Chinese and Western Medicine Shanghai University of Traditional Chinese Medicine Shanghai China.

Medcomm
|October 27, 2025
PubMed

Insights

Histone lactylation (H3K18la) drives cardiac hypertrophy by activating GATA4. Inhibiting this epigenetic modification offers a potential therapeutic strategy for hypertrophic heart diseases.

Area of Science:

  • Biochemistry
  • Epigenetics
  • Cardiovascular Biology

Background:

  • Histone lactylation, specifically H3K18la, influences gene expression and is implicated in cardiovascular disease.
  • The precise role of H3K18la in cardiac hypertrophy is not well understood.

Purpose of the Study:

  • To investigate the mechanism by which H3K18la promotes cardiac hypertrophy.
  • To explore the potential of targeting H3K18la for therapeutic interventions in hypertrophic heart disease.

Main Methods:

  • Utilized a mouse model of transverse aortic constriction and a phenylephrine-induced hypertrophic cardiomyocyte model.
  • Assessed histone lactylation levels, cardiac function markers, and gene expression.
  • Investigated the interaction between H3K18la and GATA4.

Main Results:

  • Elevated Pan-Kla and H3K18la levels were observed in hypertrophic hearts and cardiomyocytes.
  • Increased heart/left ventricle weights, cardiomyocyte size, and expression of hypertrophic markers (ANP, BNP, β-MHC) were noted.
  • H3K18la was found to interact with and enhance GATA4 transcriptional activity, which is crucial for the hypertrophic response.

Conclusions:

  • H3K18la is a novel epigenetic mechanism that promotes cardiac hypertrophy via GATA4 activation.
  • Inhibition of lactylation reversed hypertrophic effects, suggesting therapeutic potential.
  • Findings identify H3K18la and GATA4 as potential therapeutic targets for hypertrophic heart diseases.

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