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Functionalized Spirocyclic Heterocycle Synthesis and Cytotoxicity Assay
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Functionalized nitrogen- and chalcogen-containing heterocyclic compounds as aromatase inhibitors: Design, synthesis

Chang Ha Park1, Marc Le Borgne2, Marouan Rami1

  • 1Univ. Lille, Inserm, CHU Lille, U1172 - LilNCog - Lille Neuroscience & Cognition, F-59000, Lille, France.

European Journal of Medicinal Chemistry
|November 7, 2025
PubMed

Keywords:
AromataseBenzoselenazolinoneBenzothiazolinoneBenzoxazinone and benzothiazinoneBenzoxazolinoneChalcogen isostereHeterocyclesIn vitro assaysIn vivo evaluation. supplementaryNon-steroidal inhibitors

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