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Efficient Construction of Drug-like Bispirocyclic Scaffolds Via Organocatalytic Cycloadditions of α-Imino γ-Lactones and Alkylidene Pyrazolones
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Transformation of the cyclohexane ring to the cyclopentane fragment of biologically active compounds

Natalya Akhmetdinova1, Ilgiz Biktagirov2, Liliya Kh Faizullina1

  • 1Ufa Institute of Chemistry, UFRC RAS, 450054, Ufa, 71, Oktyabrya Ave. Russian Federation.

Beilstein Journal of Organic Chemistry
|November 12, 2025
PubMed

Keywords:
biological activitycyclopentane/enonerearrangementsring/cycle contractionstotal synthesis

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