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Updated: Jan 10, 2026

Parallel Interrogation of β-Arrestin2 Recruitment for Ligand Screening on a GPCR-Wide Scale using PRESTO-Tango Assay
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Parallel Interrogation of β-Arrestin2 Recruitment for Ligand Screening on a GPCR-Wide Scale using PRESTO-Tango Assay

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Noncanonical agonist-dependent and -independent arrestin recruitment of GPR1

Heng Cai1,2,3,4, Xiaowen Lin1,2,5, Lechen Zhao1,5

  • 1School of Pharmaceutical Science and Technology, Hangzhou Institute for Advanced Study, University of Chinese Academy of Sciences, Hangzhou, China.

Science (New York, N.Y.)
|November 20, 2025
PubMed

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