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Updated: Jan 8, 2026

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
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Published on: February 20, 2018

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Molecular insights into ago-allosteric modulation at cysteinyl leukotriene receptor 2

Mu Li1, Xiaoling Bao2, Wanbiao Chen3

  • 1The Affiliated Traditional Chinese Medicine Hospital, GMU-GIBH Joint School of Life Sciences, The Guangdong-Hong Kong-Macao Joint Laboratory for Cell Fate Regulation and Diseases, Guangzhou Medical University, Guangzhou Municipal and Guangdong Provincial Key Laboratory of Protein Modification and Disease, State Key Laboratory of Respiratory Disease, Guangzhou, Guangdong, China.

Nature Communications
|December 16, 2025
PubMed

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