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Published on: April 23, 2018

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Synthesis of non-steroidal cholic acid analogues as potent and selective TGR5 allosteric agonists with antidiabetic

Xinyan Shen1, Xuemei Shao1, Bowei Dong1

  • 1School of Pharmacy, Changzhou University, Changzhou 213164, PR China.

Bioorganic Chemistry
|December 27, 2025
PubMed

Keywords:
Allosteric mechanismAntidiabetic effectsScaffold hoppingTGR5 allosteric agonistsTakeda G protein coupled receptor 5

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