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Mapping ligands for MT1/MT2 and 5-HT2C receptors: Chemotypes, SAR, and polypharmacology

Alban Lepailleur1, Damien Geslin1, Johanna Giovannini1

  • 1Université Caen Normandie, Normandie Univ, CERMN UR4258, F-14000 Caen, France.

Drug Discovery Today
|January 10, 2026
PubMed
Abstract

Keywords:
5-HT(2C) serotonin receptormelatonin receptorspolypharmacologystructure–activity relationships (SARs)

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