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Asymmetric Synthesis of KRAS G12C Inhibitor MK-1084 via a Crystallization-Induced Diastereomer Transformation (CIDT)

Hongming Li1, Gao Shang1, Zhiguo J Song1

  • 1Department of Process Research and Development, Merck & Co., Inc., Rahway, New Jersey 07065, United States.

Organic Letters
|January 13, 2026
PubMed
Abstract

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