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Reducing hERG Inhibition in the Design of Potent and Bioavailable Indazole cGAS Inhibitors

Patrick Cyr1, Amandine Chefson1, Daniel V Sietsema2

  • 1Ventus Therapeutics, 4800, rue Lévy #110, Saint-Laurent, H4R 2P1 QC, Canada.

ACS Medicinal Chemistry Letters
|January 14, 2026
PubMed

Keywords:
autoimmune diseasescGAMPcGAShERGinflammation

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