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Updated: Jan 17, 2026

Characterization of G Protein-coupled Receptors by a Fluorescence-based Calcium Mobilization Assay
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Small-molecule drug discovery targeting the orphan G protein-coupled receptor GPR84 as potential therapeutics

Binghan Xue1, Yao Xiao1, Weipeng Hu2

  • 1Department of Biotherapy, State Key Laboratory of Biotherapy and Cancer Center, West China Hospital, Sichuan University, Chengdu, 610041, China.

European Journal of Medicinal Chemistry
|January 14, 2026
PubMed

Keywords:
AgonistsAntagonistsDiseasesGPCRGPR84Structure-activity relationship

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