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Updated: Jun 17, 2026

Incorporating Target Protein Structure Flexibility and Dynamics in Computational Drug Discovery Using Ensemble-Based Docking Analysis
Published on: June 20, 2025
J O Lannot1,2, E L Rey1,2, M D Gamarra1,2
1Departamento de Química Biológica, Facultad de Ciencias Exactas y Naturales, Universidad de Buenos Aires (FCEyN-UBA), Pabellón 2 de Ciudad Universitaria, Ciudad de Buenos Aires C1428EHA, Buenos Aires, Argentina.
We developed a guided docking protocol using crystallographic water sites (CWS) to improve protein-carbohydrate complex structure prediction. This novel approach enhances glycan pose prediction accuracy for drug discovery.
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