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Design, synthesis, and biological evaluation of hydrophobic-tagged poly (ADP-ribose) polymerase 1 (PARP1) degraders

Jiaqian Li1, Yang Cui2, Mengyu Xiong3

  • 1School of Pharmacy, North China University of Science and Technology, Tangshan 063210, China.

Bioorganic Chemistry
|January 21, 2026
PubMed

Keywords:
CancerDegradationHydrophobic taggingPARP1

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