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Updated: Jan 29, 2026

Quantifying Agonist Activity at G Protein-coupled Receptors
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Quantifying Agonist Activity at G Protein-coupled Receptors

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Improved synthesis and physicochemical characterization of the selective serotonin 2A receptor agonist 25CN-NBOH

Adrian G Rossebø1, Hannah G Kolberg2,3, Anders E Tønder1

  • 1Department of Drug Design and Pharmacology, Faculty of Health and Medical Sciences, University of Copenhagen, Jagtvej 162, 2100 Copenhagen, Denmark.

Beilstein Journal of Organic Chemistry
|January 28, 2026
PubMed

Keywords:
intramolecular hydrogen bondmembrane permeabilitysolubilitystabilitysynthesis

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