A dialogue on innovation in anticancer drug discovery

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Updated: Feb 5, 2026

Assessing Specificity of Anticancer Drugs In Vitro
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Assessing Specificity of Anticancer Drugs In Vitro

Published on: March 23, 2016

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Susanta Samajdar1

  • 1Aurigene Oncology Limited 39-40, KIADB Industrial Area, Electronic City Phase II, Hosur Road Bangalore - 560100 India susanta_s@aurigene.com.

RSC Medicinal Chemistry
|February 4, 2026
PubMed

Insights

Medicinal chemistry has advanced cancer drug discovery from chemotherapy to precision therapies. Emerging innovations like proximity inducers and drug conjugates offer new hope but require overcoming delivery and resistance challenges.

Area of Science:

  • Medicinal Chemistry
  • Oncology Drug Discovery
  • Cancer Therapeutics

Background:

  • The evolution of oncology drug discovery is marked by medicinal chemistry's pivotal role.
  • Early cytotoxic agents have been succeeded by sophisticated precision-guided therapies.
  • This progression reflects advancements in understanding cancer biology and drug development.

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