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Updated: Feb 7, 2026

Microwave-Assisted Preparation of 1-Aryl-1H-pyrazole-5-amines
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Structure-Based Design of 4-(1-Methyl-1H-indol-3-yl)pyrimidin-2-amine Derivatives as the First Covalent FGFR3

Wenjian Zhu1, Xiaojuan Chen2, Xiaofei Li1

  • 1State Key Laboratory of Bioactive Molecules and Druggability Assessment, Guangdong Basic Research Center of Excellence for Natural Bioactive Molecules and Discovery of Innovative Drugs, International Cooperative Laboratory of Traditional Chinese Medicine Modernization and Innovative Drug Discovery of Chinese Ministry of Education, Guangzhou City Key Laboratory of Precision Chemical Drug Development, School of Pharmacy, Jinan University, Guangzhou 510632, China.

Journal of Medicinal Chemistry
|February 6, 2026
PubMed

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