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Updated: Feb 19, 2026

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Synthesis and Biological Evaluation of 3,5-Diaryl-Substituted 1,2,4-Oxadiazole Sulfamates as Potent Steroid Sulfatase

Karol Biernacki1, Olga Ciupak2, Mateusz Daśko2

  • 1Department of Organic Chemistry, Faculty of Chemistry, Gdańsk University of Technology, Narutowicza 11/12 Street, 80-233 Gdańsk, Poland.

ACS Medicinal Chemistry Letters
|February 18, 2026
PubMed

Keywords:
1,2,4-oxadiazoleSteroid sulfatasebreast cancerdrug designmolecular modelingstructure−activity relationship

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