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Updated: Feb 20, 2026

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Enantioselective S-Alkylation of Sulfenamides With Copper-Catalyzed Amino-Radical-Transfer Deboronation

Ke Wang1, Yu Qi1, Menghui Ding1

  • 1Department of Medicinal Chemistry, State Key Laboratory of Discovery and Utilization of Functional Components in Traditional Chinese Medicine, Shandong Key Laboratory of Druggability Optimization and Evaluation for Lead Compounds, School of Pharmaceutical Sciences, Shandong University, Jinan, Shandong, China.

Angewandte Chemie (International Ed. in English)
|February 18, 2026
PubMed

Keywords:
asymmetric alkylationchiral sulfiliminecopper catalysisdeboronationradical relay coupling

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