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Updated: May 12, 2026

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
07:41

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Assessment of high-efficacy agonism in synthetic cannabinoid receptor agonists containing l-tert-leucinate

Christopher Lucaj1, Soo Jung Oh1, Charlotte Pitha1

  • 1Department of Pharmaceutical Sciences, School of Pharmacy and Pharmaceutical Sciences, Bouvé College of Health Sciences, Center for Drug Discovery, Northeastern University, Boston, MA, 02115, United States.

Neuropharmacology
|February 19, 2026
PubMed

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