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Updated: Feb 22, 2026

Methods for the Discovery of Novel Compounds Modulating a Gamma-Aminobutyric Acid Receptor Type A Neurotransmission
07:16

Methods for the Discovery of Novel Compounds Modulating a Gamma-Aminobutyric Acid Receptor Type A Neurotransmission

Published on: August 16, 2018

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Recent advances in GABAA receptor targeting ligands

Yuanyan Zuo1, Yilan Zhao2, Genyan Liu1

  • 1Hubei Key Laboratory of Novel Reactor and Green Chemical Technology, Key Laboratory for Green Chemical Process of Ministry of Education, School of Chemical Engineering and Pharmacy, Wuhan Institute of Technology, Wuhan, 430205, PR China.

European Journal of Medicinal Chemistry
|February 20, 2026
PubMed
Abstract

Keywords:
Allosteric modulatorsCryo-EM structuresGABA(A) receptorNeuropsychiatric disordersStructure-based drug designSubtype selectivity

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