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Updated: Feb 28, 2026

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
07:41

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators

Published on: February 20, 2018

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Structural determinants for GPCR-mediated inhibition of TASK K2P channels by diacylglycerol and its dysfunction in

Thibault R H Jouen-Tachoire1,2,3,4, Peter Proks1,2, David Seiferth5,2

  • 1Kavli Institute for Nanoscience Discovery, University of Oxford, Oxford, UK.

The EMBO Journal
|February 25, 2026
PubMed

Keywords:
ChannelopathyDiacylglycerolGPCR/K2P ChannelKCNK3

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