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Optimization of α-Fluoro, β-Heteroaryl Acrylamide Warheads for KRASG12C Active-State Inhibition

Matthew L Condakes1, Rita L Civiello1, Brian L Venables1

  • 1Bristol Myers Squibb, 250 Water St., Cambridge, Massachusetts 02446, United States.

Journal of Medicinal Chemistry
|March 2, 2026
PubMed

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