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Discovery of Potent and Brain-Penetrant Inverse Agonists for GPR61, an Orphan G Protein-Coupled Receptor

Ethan L Fisher1, Anne-Marie Dechert Schmitt1, Jamison B Tuttle2

  • 1Pfizer Research & Development, 558 Eastern Point Rd, Groton, Connecticut 06340, United States.

Journal of Medicinal Chemistry
|March 16, 2026
PubMed
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