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Methods for the Discovery of Novel Compounds Modulating a Gamma-Aminobutyric Acid Receptor Type A Neurotransmission
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6,7-Dihalo-Benzothiadiazines as Potent and Selective AMPA Receptor Modulators for Cognitive Enhancement and

Yinlong Li1, Hongjie Yuan2, Steven H Liang1,3

  • 1Department of Radiology and Imaging Sciences, Emory University, 1364 Clifton Road, Atlanta, Georgia 30322, United States.

ACS Medicinal Chemistry Letters
|March 18, 2026
PubMed

Keywords:
AMPA receptorNeurological disordersPositive allosteric modulatorsStructure−activity relationship

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