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Updated: Mar 24, 2026

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Insights Into Vepdegestrant (ARV-471): The First-in-Class Estrogen Receptor Proteolysis-Targeting Chimera Approaching

Chao Tang1,2, Bin Tian1,2, Bingxing Zhang1,2

  • 1School of Biological and Pharmaceutical Sciences, Shaanxi University of Science & Technology, Weiyang University Park, Xi'an, Shaanxi, China.

Chemmedchem
|March 23, 2026
PubMed

Keywords:
breast cancerestrogen receptor degraderproteolysis‐targeting chimeratargeted protein degradationvepdegestrant (ARV‐471)

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