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Unravelling Structure-Based Molecular Activation and Antagonism of Protease-Activated Receptors for Drug Design

Zhikang Xu1, Rui Li1, Jian Zhang1,2,3

  • 1Artificial Intelligence Clinical Research Center for Drug Discovery, Shanghai Key Laboratory of Flexible Medical Robotics, Tongren Hospital, Shanghai Jiao Tong University School of Medicine, Shanghai, China.

Medicinal Research Reviews
|April 3, 2026
PubMed

Keywords:
activationallosteric modulatorligand recognitionprotease‐activated receptorstructure

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