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Updated: May 8, 2026

Preparation of Stable Bicyclic Aziridinium Ions and Their Ring-Opening for the Synthesis of Azaheterocycles
11:45

Preparation of Stable Bicyclic Aziridinium Ions and Their Ring-Opening for the Synthesis of Azaheterocycles

Published on: August 22, 2018

Strain Release of 1-Azabicyclo[1.1.0]butanes as a Gateway to Highly Functionalized Azetidines: New Strategies and

Yuri Gelato1, Philipp Natho1, Marco Colella1

  • 1Department of Pharmacy-Drug Sciences, University of Bari "A. Moro", Bari, Italy.

Chemistry (Weinheim an Der Bergstrasse, Germany)
|May 7, 2026
PubMed

Keywords:
1‐azabicyclo[1.1.0]butanesazetidinesbioisosteresspirocyclestechnologies

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