Related Experiment Video

Updated: May 31, 2026

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
07:41

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators

Published on: February 20, 2018

Kainate Receptor Allosteric Modulators: State of the Art and Future Directions

Thomas Colson1, Bernard Pirotte1, Pierre Francotte1

  • 1Laboratory of Medicinal Chemistry, CIRM, Department of Pharmacy, University of Liège, Liège, Belgium.

Chemmedchem
|May 29, 2026
PubMed
Abstract

Keywords:
allosteric modulationkainate receptorspositive and negative modulatorsstructure‐guided drug designsubunit selectivity

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