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Updated: Jun 13, 2026

Methods for the Discovery of Novel Compounds Modulating a Gamma-Aminobutyric Acid Receptor Type A Neurotransmission
07:16

Methods for the Discovery of Novel Compounds Modulating a Gamma-Aminobutyric Acid Receptor Type A Neurotransmission

Published on: August 16, 2018

First Structure-Activity-Relationship Study of Potent G2A Antagonists

Victor Hernandez-Olmos1,2, Jan Heering1,2, Felix F Lillich3

  • 1Fraunhofer Institute for Translational Medicine and Pharmacology ITMP, Theodor-Stern-Kai 7, 60596 Frankfurt am Main, Germany.

Journal of Medicinal Chemistry
|June 11, 2026
PubMed

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